الصفحة الرئيسية

كلية الصيدلة \ الكيمياء الصيدلة

نادر المغاوري مصطفى أبوديه

نسبة اكتمال الملف الشخصي
الجنسية المصرية
التخصص العام الكيمياء الصيدلية
التخصص الدقيق الكيمياء العضوية الصيدلية
المسمى الوظيفي أستاذ مساعد
الدرجة العلمية (المرتبة) دكتوراه

نبذه مختصرة

 Profile  A highly motivated and competent Pharmaceutical chemist  Associate Professor of Organic and medicinal chemistry  Ten years of teaching pharmaceutical Organic Chemistry courses to  both graduate and undergraduate pharmacy students at University of  Tabuk (Saudi Arabia), Zagazig University , Misr International University,  and Delta University of Science and Technology (Egypt)  Five years of Teaching Medicinal Chemistry courses and Drug design at the Faculty of Pharmacy, University of Tabuk, KSA --Two Years of experience as a research scholar at the Department of --Chemistry, University of Florida, USA under supervision of Prof Alan Roy Katritzky --One year as Postdoc and Group leader at the Center of Heterocyclic --Compounds, Department of Chemistry, University of Florida, USA --Visiting scholar at the Department of Chemistry, King Abdul-Aziz --University, Jeddah, and KSA (August-September 2012) --Visiting professor at Oman College of health sciences (school of Pharmacy), Muscat, Oman (September -December 2014) --Over 6 years of experience as a teaching assistant at Zagazig University --Member of the ACS and the RSC

المؤهلات العلمية

PhD in Pharmaceutical Organic Chemistry - Faculty of Pharmacy - Zagazig University - Egypt - Joint Supervision with University of Florida, USA - 2010 Master in Pharmaceutical Organic Chemistry - Faculty of Pharmacy - Zagazig University - Egypt - 2006 1999- Bachelor of Pharmaceutical Sciences - Faculty of Pharmacy - Zagazig University - Egypt

الاهتمامات البحثية

Peptidomimetics Benzotriazole as a synthetic auxillary Chemotherapeutic agents Drugs for neurodegenerative disorders and cognitive enhancers Design and synthesis of anticancer protein kinase inhibitors

الخبرات والمناصب الإدارية

Head of Pharmaceutical Chemistry Department - Faculty of Pharmacy- University of Tabuk 2017-to present Supervisor of Evaluation and Assessment Unit at Faculty of Pharmacy- University of Tabuk 2018-2020

الجدول الدراسي
اليوم المادة الوقت
من إلى
الأحد Pharmaceutical Analytical chemistry- Male students 09:00 12:00
الأحد Office hours male students 12:00 13:00
الإثنين Pharmaceutical Organic Chemistry-Male students 08:00 10:00
الإثنين Academic Advising 11:00 12:00
الإثنين Office hours male students 12:00 13:00
الثلاثاء Pharmaceutical Organic Chemistry-Female students 09:00 12:00
الثلاثاء Office hours female students 12:00 15:00
الأربعاء Pharmaceutical Organic Chemistry-Male students 08:00 09:00
الأربعاء Office hours male students 12:00 13:00
الخميس Pharmaceutical Field Training-3- Male 08:00 12:00
الخميس Academic Advising 12:00 13:00
الأبحاث والمؤلفات
  • Design, synthesis and pharmacological screening of novel renoprotective methionine-based peptidomimetics: Amelioration of cisplatin-induced nephrotoxicity Bioorganic Chemistry 2021 | journal-article DOI: 101016/jbioorg2021105100EID: 2-s20-85109456295Part of ISSN: 10902120 00452068
  • Design, synthesis and anticancer activity of novel valproic acid conjugates with improved histone deacetylase (HDAC) inhibitory activity Bioorganic Chemistry 2020 | journal-article DOI: 101016/jbioorg2020103797EID: 2-s20-85082706397Part of ISSN: 10902120 00452068
  • N-Acylbenzotriazole: convenient approach for protecting group-free monoacylation of symmetric diamines Monatshefte fur Chemie 2020 | journal-article DOI: 101007/s00706-020-02579-5EID: 2-s20-85084154007Part of ISSN: 00269247
  • Benzotriazole-mediated synthesis and antibacterial activity of novel n-acylcephalexins Scientia Pharmaceutica 2016 | journal-article DOI: 103390/scipharm84030484EID: 2-s20-84992053084Part of ISSN: 22180532 00368709
  • Efficient synthesis of N-acylbenzotriazoles using tosyl chloride: En route to suberoylanilide hydroxamic acid (SAHA) Arkivoc 2016 | journal-article DOI: 103998/ark5550190p009459EID: 2-s20-84975137669Part of ISSN: 15517012 15517004
  • Benzotriazole-mediated synthesis of aza-peptides: En route to an aza-leuenkephalin analogue Journal of Organic Chemistry 2013 | journal-article DOI: 101021/jo302251eEID: 2-s20-84876583019Part of ISSN: 00223263 15206904
  • Non-phosgene route to unsymmetrical ureas from N-Cbz-α-amino acid amides Tetrahedron Letters 2013 | journal-article DOI: 101016/jtetlet201307141EID: 2-s20-84883453537Part of ISSN: 00404039 18733581
  • Oxyazapeptides: Synthesis, structure determination, and conformational analysis Journal of Organic Chemistry 2013 | journal-article DOI: 101021/jo401234gEID: 2-s20-84883827766Part of ISSN: 00223263 15206904
  • Photophysics of novel coumarin-labeled depsipeptides in solution: Sensing interactions with SDS micelle via TICT model Amino Acids 2013 | journal-article DOI: 101007/s00726-013-1483-3EID: 2-s20-84879224868Part of ISSN: 09394451 14382199
  • 1-(1H-1,2,3-Benzotriazol-1-yl)-2-(4-methoxyphenyl)ethanone Acta Crystallographica Section E: Structure Reports Online 2012 | journal-article DOI: 101107/S1600536812043759 https://doiorg/101107/s1600536812043759 EID: 2-s20-84870895907Part of ISSN: 16005368
  • 1-(Benzotriazol-1-yl)-2-bromoethanone Acta Crystallographica Section E: Structure Reports Online 2012 | journal-article DOI: 101107/S1600536812042900EID: 2-s20-84870904274Part of ISSN: 16005368
  • Chemical ligation of S-scylated cysteine peptides to form native peptides via 5-, 11-, and 14-membered cyclic transition states Journal of Organic Chemistry 2011 | journal-article DOI: 101021/jo1015757EID: 2-s20-78650874855Part of ISSN: 00223263 15206904
  • DBU-Catalyzed transprotection of N-Fmoc-cysteine di- and tripeptides into S-Fm-cysteine di- and tripeptides Organic and Biomolecular Chemistry 2011 | journal-article DOI: 101039/c0ob00663gEID: 2-s20-78650733758Part of ISSN: 14770520
  • Design, synthesis, and biological activity of a novel series of 2,5-disubstituted furans/pyrroles as HIV-1 fusion inhibitors targeting gp41 Bioorganic and Medicinal Chemistry Letters 2011 | journal-article DOI: 101016/jbmcl201108081EID: 2-s20-80054723128Part of ISSN: 0960894X 14643405
  • Design, synthesis, and biological activity of novel 5-((arylfuran/1 H -pyrrol-2-yl)methylene)-2-thioxo-3-(3-(trifluoromethyl)phenyl) thiazolidin-4-ones as HIV-1 fusion inhibitors targeting gp41 Journal of Medicinal Chemistry 2011 | journal-article DOI: 101021/jm101014vEID: 2-s20-78751657690Part of ISSN: 00222623 15204804
  • Synthesis of coumarin conjugates of biological thiols for fluorescent detection and estimation Synthesis 2011 | journal-article DOI: 101055/s-0030-1259991EID: 2-s20-79955022459Part of ISSN: 00397881 1437210X
  • Efficient and selective syntheses of S -Acyl and N -Acyl glutathiones Synlett 2010 | journal-article DOI: 101055/s-0029-1219837EID: 2-s20-77953281405Part of ISSN: 09365214 14372096
  • The chemical ligation of selectively S-acylated cysteine peptides to form native peptides via 5-, 11- and 14-membered cyclic transition states Organic and Biomolecular Chemistry 2010 | journal-article DOI: 101039/c003234dEID: 2-s20-77952364392Part of ISSN: 14770520
  • An efficient method for the preparation of peptide alcohols Organic and Biomolecular Chemistry 2009 | journal-article DOI: 101039/b905730gEID: 2-s20-70350007193Part of ISSN: 14770520
  • Efficient synthesis of azo dye labeled terpenes, sugars, and steroids using N-(4-arylazobenzoyl)-1H-benzotriazoles Synthesis 2009 | journal-article DOI: 101055/s-0029-1216786EID: 2-s20-67650021159Part of ISSN: 00397881 1437210X
  • Selective synthesis and structural elucidation of S-acyl- and N-acylcysteines Journal of Organic Chemistry 2009 | journal-article DOI: 101021/jo900853sEID: 2-s20-70249129814Part of ISSN: 00223263
  • Photophysics of novel coumarin-labeled depsipeptides in solution: sensing interactions with SDS micelle via TICT model S Biswas, I Avan, AK Basak, NE Abo-Dya, A Asiri, AR Katritzky Amino acids 45 (1), 159-170
  • Peptide hydroxamate derivatives as regulators for insulin receptor signaling and its degradation by zinc metalloprotease in diabetic rats MM Elseweidy, RS Amin, HH Atteia, MA Ali, NE Abo-Dya, KA Agha African Journal of Pharmacy and Pharmacology 10 (30), 616-622
  • Propitious Indazole Compounds as β‐ketoacyl‐ACP Synthase Inhibitors and Mechanisms Unfolded for TB Cure: Integrated Rational Design and MD Simulations‏ AT Adewumi, WM Oluyemi, YA Adekunle, N Adewumi, MI Alahmdi, NE Abo-Dya, ‏ ChemistrySelect 8 (3), e202203877
  • Revealing the Role of the Arg and Lys in Shifting Paradigm from BTK Selective inhibition to the BTK/HCK Dual inhibition-Delving into the Inhibitory Activity of KIN-8194 Against …‏ G Elamin, A Aljoundi, M Alahmdi, NE Abo-Dya, M Soliman NE Abo-Dya, ‏‏ Anti-cancer Agents in Medicinal Chemistry‏2023
جوائز التميز
  • Best PhD Thesis from Zagazig University 2010
  • جائزة التميز في التدريس كلية الصيدلة -جامعة تبوك-1444هـ
المشاريع البحثية
اسم المشروع وصف المشروع
Design, Synthesis and Biological Studies of Novel pyrazoline and moracin based compounds as antihyperglycemic agents and aldose reductase inhibitors Submitted for acceptance by the deanship of scientific research
معلومات التواصل
البريد الإلكتروني : nabodya@ut.edu.sa
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